BI-D1870 : MKNK1 is a YB-1 target gene responsible for imparting trastuzumab resistance and can be blocked by RSK inhibition

GSK343: Novel strategies for molecular targeting to cancer

LLY-283 : Discovery and Mechanistic Study of a Class of Protein Arginine Methylation Inhibitors

Tucatinib : Prevention of brain metastases in human epidermal growth factor receptor 2-positive breast cancer

AGI-6780 : IDH2 mutation-induced histone and DNA hypermethylation is progressively reversed by small-molecule inhibition